Tiziano Tuccinardi
Tiziano Tuccinardi
Associate Professor, University of Pisa
Verified email at unipi.it - Homepage
Title
Cited by
Cited by
Year
Discovery of N-Hydroxyindole-Based Inhibitors of Human Lactate Dehydrogenase Isoform A (LDH-A) as Starvation Agents against Cancer Cells
C Granchi, S Roy, C Giacomelli, M Macchia, T Tuccinardi, A Martinelli, ...
Journal of medicinal chemistry 54 (6), 1599-1612, 2011
1852011
Cannabinoid CB2/CB1 selectivity. Receptor modeling and automated docking analysis
T Tuccinardi, PL Ferrarini, C Manera, G Ortore, G Saccomanni, ...
Journal of medicinal chemistry 49 (3), 984-994, 2006
1252006
Matrix metalloproteinase inhibitors: new challenges in the era of post broad-spectrum inhibitors
E Nuti, T Tuccinardi, A Rossello
Current pharmaceutical design 13 (20), 2087-2100, 2007
1132007
CDK inhibitors: from the bench to clinical trials
F Rizzolio, T Tuccinardi, I Caligiuri, C Lucchetti, A Giordano
Current drug targets 11 (3), 279-290, 2010
942010
Docking-based virtual screening: recent developments
T Tuccinardi
Combinatorial chemistry & high throughput screening 12 (3), 303-314, 2009
882009
Amber force field implementation, molecular modelling study, synthesis and MMP-1/MMP-2 inhibition profile of (R)- and (S)-N-hydroxy-2-(N-isopropoxybiphenylá…
T Tuccinardi, A Martinelli, E Nuti, P Carelli, F Balzano, G Uccello-Barretta, ...
Bioorganic & medicinal chemistry 14 (12), 4260-4276, 2006
852006
Proposal of a new binding orientation for non-peptide AT1 antagonists: Homology modeling, docking and three-dimensional quantitative structure− activity relationship analysis
T Tuccinardi, V Calderone, S Rapposelli, A Martinelli
Journal of medicinal chemistry 49 (14), 4305-4316, 2006
822006
Targeting toxic RNAs that cause myotonic dystrophy type 1 (DM1) with a bisamidinium inhibitor
CH Wong, L Nguyen, J Peh, LM Luu, JS Sanchez, SL Richardson, ...
Journal of the American Chemical Society 136 (17), 6355-6361, 2014
812014
New 1, 8-naphthyridine and quinoline derivatives as CB2 selective agonists
C Manera, MG Cascio, V Benetti, M AllarÓ, T Tuccinardi, A Martinelli, ...
Bioorganic & medicinal chemistry letters 17 (23), 6505-6510, 2007
772007
Design, synthesis, and biological evaluation of new 1, 8-naphthyridin-4 (1 H)-on-3-carboxamide and quinolin-4 (1 H)-on-3-carboxamide derivatives as CB2 selective agonists
C Manera, V Benetti, MP Castelli, T Cavallini, S Lazzarotti, F Pibiri, ...
Journal of medicinal chemistry 49 (20), 5947-5957, 2006
742006
Protein kinases: docking and homology modeling reliability
T Tuccinardi, M Botta, A Giordano, A Martinelli
Journal of chemical information and modeling 50 (8), 1432-1441, 2010
662010
The TRPA 1 channel mediates the analgesic action of dipyrone and pyrazolone derivatives
R Nassini, C Fusi, S Materazzi, E Coppi, T Tuccinardi, IM Marone, ...
British journal of pharmacology 172 (13), 3397-3411, 2015
642015
N-Hydroxyindole-based inhibitors of lactate dehydrogenase against cancer cell proliferation
C Granchi, S Roy, A De Simone, I Salvetti, T Tuccinardi, A Martinelli, ...
European journal of medicinal chemistry 46 (11), 5398-5407, 2011
642011
Derivatives of 4-Amino-6-hydroxy-2-mercaptopyrimidine as Novel, Potent, and Selective A3 Adenosine Receptor Antagonists
B Cosimelli, G Greco, M Ehlardo, E Novellino, F Da Settimo, S Taliani, ...
Journal of medicinal chemistry 51 (6), 1764-1770, 2008
602008
Extensive consensus docking evaluation for ligand pose prediction and virtual screening studies
T Tuccinardi, G Poli, V Romboli, A Giordano, A Martinelli
Journal of chemical information and modeling 54 (10), 2980-2986, 2014
592014
Molecular modeling of adenosine receptors: new results and trends
A Martinelli, T Tuccinardi
Medicinal research reviews 28 (2), 247-277, 2008
582008
N-O-Isopropyl Sulfonamido-Based Hydroxamates: Design, Synthesis and Biological Evaluation of Selective Matrix Metalloproteinase-13 Inhibitors as Potentialá…
E Nuti, F Casalini, SI Avramova, S Santamaria, G Cercignani, L Marinelli, ...
Journal of medicinal chemistry 52 (15), 4757-4773, 2009
542009
Indoles and related compounds as cannabinoid ligands
C Manera, T Tuccinardi, A Martinelli
Mini reviews in medicinal chemistry 8 (4), 370-387, 2008
522008
α-Glucosidase and α-Amylase Inhibitors from Arcytophyllum thymifolium
L Milella, S Milazzo, M De Leo, MB Vera Saltos, I Faraone, T Tuccinardi, ...
Journal of Natural Products 79 (8), 2104-2112, 2016
512016
Assessing the differential action on cancer cells of LDH-A inhibitors based on the N-hydroxyindole-2-carboxylate (NHI) and malonic (Mal) scaffolds
C Granchi, EC Calvaresi, T Tuccinardi, I Paterni, M Macchia, A Martinelli, ...
Organic & biomolecular chemistry 11 (38), 6588-6596, 2013
512013
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